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Trial details imported from ClinicalTrials.gov

For full trial details, please see the original record at https://clinicaltrials.gov/study/NCT01820364




Registration number
NCT01820364
Ethics application status
Date submitted
25/03/2013
Date registered
28/03/2013
Date last updated
9/01/2017

Titles & IDs
Public title
LGX818 in Combination With Agents (MEK162; BKM120; LEE011; BGJ398; INC280) in Advanced BRAF Melanoma
Scientific title
Phase II, Multi-center, Open-label Study of Single-agent LGX818 Followed by a Rational Combination With Agents After Progression on LGX818, in Adult Patients With Locally Advanced or Metastatic BRAF V600 Melanoma
Secondary ID [1] 0 0
2012-004798-17
Secondary ID [2] 0 0
CLGX818X2102
Universal Trial Number (UTN)
Trial acronym
LOGIC
Linked study record

Health condition
Health condition(s) or problem(s) studied:
Melanoma 0 0
Condition category
Condition code
Cancer 0 0 0 0
Malignant melanoma

Intervention/exposure
Study type
Interventional
Description of intervention(s) / exposure
Treatment: Drugs - LGX818

Experimental: LGX818 single agent - Patients had to have written documentation of a BRAFV600 mutation, which was to have been obtained locally on a fresh tumor biopsy (preferred) or on the most recent archival tumor sample available.


Treatment: Drugs: LGX818
BRAF inhibitor. LGX818 was administered QD orally on a daily schedule (21-day cycles) as a flat-fixed dose and not by body weight or body surface area. LGX818 100 mg capsules and 50 mg capsules.

Intervention code [1] 0 0
Treatment: Drugs
Comparator / control treatment
Control group

Outcomes
Primary outcome [1] 0 0
Tumor Response (Overall Response Rate) Per Response Evaluation Criteria In Solid Tumors (RECIST) v1.1 (Part I & Part II)
Timepoint [1] 0 0
Baseline through study completion (approximately 2 years)
Secondary outcome [1] 0 0
Incidence of Dose Limiting Toxicities (DLTs) (Part II)
Timepoint [1] 0 0
Baseline through study completion (approximately 2 years)
Secondary outcome [2] 0 0
Plasma Concentration and Derived Pharmacokinetic Parameters
Timepoint [2] 0 0
Baseline through study completion (approximately 2 years)
Secondary outcome [3] 0 0
Tumor Response (Overall Response Rate) Via Response Evaluation Criteria In Solid Tumors (RECIST) v1.1 (Part I)
Timepoint [3] 0 0
Baseline through completion of Part I of the study (approximately 2 years)
Secondary outcome [4] 0 0
Tumor Response (Overall Response Rate) Via Response Evaluation Criteria In Solid Tumors (RECIST) v1.1 (Part II)
Timepoint [4] 0 0
Entry to Part II of the study through study completion (approximately 22 days)
Secondary outcome [5] 0 0
Molecular Status of Markers Relevant to the RAP/MEK/ERK and PI3K/AKT Pathways
Timepoint [5] 0 0
Baseline and at progression with LGX818 single agent treatment

Eligibility
Key inclusion criteria
* locally advanced or metastatic melanoma
* confirmed BRAF V600 mutation
* patients naïve to a selective BRAF inhibitor
* fresh tumor biopsy at baseline, and patient agrees for a mandatory biopsy at the time of relapse
* life expectancy = 3 months
* World Health Organization (WHO) Performance Status = 2.
Minimum age
18 Years
Maximum age
No limit
Sex
Both males and females
Can healthy volunteers participate?
No
Key exclusion criteria
* Previous treatment with RAF-inhibitor
* Symptomatic or untreated leptomeningeal disease
* Symptomatic brain metastases.
* Known acute or chronic pancreatitis
* Clinically significant cardiac disease
* AST/SGOT and ALT/SGPT > 2.5 x ULN, or > 5 x ULN if liver metastases are present
* Impairment of gastrointestinal (GI) function or GI disease that may significantly alter the absorption of oral interventional drug
* Previous or concurrent malignancy.
* Other severe, acute, or chronic medical or psychiatric condition or laboratory abnormality that may increase the risk associated with study participation

Specific exclusion criteria for each treatment arm:

LGX818/MEK162:

History or current evidence of retinal disease History of Gilbert's syndrome.

LGX818/BKM120:

Patients with diabetes mellitus requiring insulin treatment Patient has mood disorders

LGX818/BGJ398:

History and/or current evidence of ectopic mineralization/ calcification Current evidence of corneal disorder/ keratopathy Patients with current evidence of endocrine alteration of calcium/phosphate homeostasis.

History of congenital long QT- syndrome and/or hypokalaemia CTCAE Grade = 3 and/or magnesium levels below the clinically relevant lower limits before study entry.

Ionized (i) calcium (Ca) > ULN Serum inorganic phosphorus (Pi) > ULN

LGX818/LEE011 History of congenital long QT- syndrome and/or hypokalaemia CTCAE Grade = 3 and/or magnesium levels below the clinically relevant lower limits before study entry.

Study design
Purpose of the study
Treatment
Allocation to intervention
NA
Procedure for enrolling a subject and allocating the treatment (allocation concealment procedures)
Methods used to generate the sequence in which subjects will be randomised (sequence generation)
Masking / blinding
Open (masking not used)
Who is / are masked / blinded?



Intervention assignment
Single group
Other design features
Phase
Phase 2
Type of endpoint/s
Statistical methods / analysis

Recruitment
Recruitment status
Stopped early
Data analysis
Reason for early stopping/withdrawal
Other reasons
Date of first participant enrolment
Anticipated
Actual
Date of last participant enrolment
Anticipated
Actual
Date of last data collection
Anticipated
Actual
Sample size
Target
Accrual to date
Final
Recruitment in Australia
Recruitment state(s)
VIC
Recruitment hospital [1] 0 0
Novartis Investigative Site - East Melbourne
Recruitment postcode(s) [1] 0 0
3002 - East Melbourne
Recruitment outside Australia
Country [1] 0 0
United States of America
State/province [1] 0 0
Tennessee
Country [2] 0 0
Canada
State/province [2] 0 0
Alberta
Country [3] 0 0
Germany
State/province [3] 0 0
Heidelberg
Country [4] 0 0
Spain
State/province [4] 0 0
Catalunya
Country [5] 0 0
Switzerland
State/province [5] 0 0
Zuerich

Funding & Sponsors
Primary sponsor type
Commercial sector/industry
Name
Array BioPharma
Address
Country

Ethics approval
Ethics application status

Summary
Brief summary
Trial website
Trial related presentations / publications
Public notes

Contacts
Principal investigator
Name 0 0
Array BioPharma
Address 0 0
303-381-6604
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for public queries
Name 0 0
Address 0 0
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for scientific queries

No information has been provided regarding IPD availability


What supporting documents are/will be available?

No Supporting Document Provided



Results publications and other study-related documents

No documents have been uploaded by study researchers.