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Trial details imported from ClinicalTrials.gov

For full trial details, please see the original record at https://clinicaltrials.gov/study/NCT03384290




Registration number
NCT03384290
Ethics application status
Date submitted
26/11/2017
Date registered
27/12/2017

Titles & IDs
Public title
Study of a Single Dose of PRS-060 Administered by Oral Inhalation or IV Infusion in Healthy Subjects
Scientific title
A Dose Escalating Single Blind Study to Assess the Safety, Tolerability and Pharmacokinetics of a Single Dose of PRS-060 Administered by Oral Inhalation or IV Infusion in Healthy Subjects
Secondary ID [1] 0 0
PRS-060-PCS_06_17
Universal Trial Number (UTN)
Trial acronym
Linked study record

Health condition
Health condition(s) or problem(s) studied:
Healthy Subjects 0 0
Condition category
Condition code
Respiratory 0 0 0 0
Other respiratory disorders / diseases

Intervention/exposure
Study type
Interventional
Description of intervention(s) / exposure
Treatment: Drugs - PRS-060
Treatment: Drugs - Placebo

Placebo comparator: Placebo -

Experimental: PRS-060 -


Treatment: Drugs: PRS-060
Drug

Treatment: Drugs: Placebo
PRS-060 Matching Placebo

Intervention code [1] 0 0
Treatment: Drugs
Comparator / control treatment
Control group

Outcomes
Primary outcome [1] 0 0
Number of participants with Adverse Events (AEs) after a single inhaled or IV infusion dose of PRS-060.
Timepoint [1] 0 0
From time of dose until 30 days after dosing.
Primary outcome [2] 0 0
Change in blood pressure.
Timepoint [2] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [3] 0 0
Change in heart rate.
Timepoint [3] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [4] 0 0
Change in body temperature.
Timepoint [4] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [5] 0 0
Change in electrocardiograms (ECGs).
Timepoint [5] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [6] 0 0
Change in FEV1 (Forced expiratory volume 1-second)
Timepoint [6] 0 0
Pre-dose and post-dose at 5,10, 20 minutes,1 and 4 hours
Primary outcome [7] 0 0
Change in FEV6 (Forced expiratory volume 6-seconds)
Timepoint [7] 0 0
Pre-dose and post-dose at 5, 10, 20 minutes,1 and 4 hours
Primary outcome [8] 0 0
Change in peak expiratory flow rate (PEFR)
Timepoint [8] 0 0
Pre-dose and post-dose at 5, 10, 20 minutes,1 and 4 hours
Primary outcome [9] 0 0
Change in forced vital capacity (FVC)
Timepoint [9] 0 0
Pre-dose and post-dose at 5, 10, 20 minutes,1 and 4 hours
Primary outcome [10] 0 0
Change in sodium levels as part of standard serum chemistry panel.
Timepoint [10] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [11] 0 0
Change in potassium levels as part of standard serum chemistry panel.
Timepoint [11] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [12] 0 0
Change in chloride levels as part of standard serum chemistry panel.
Timepoint [12] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [13] 0 0
Change in bicarbonate levels as part of standard serum chemistry panel.
Timepoint [13] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [14] 0 0
Change in blood urea nitrogen (BUN) / Urea levels as part of standard serum chemistry panel.
Timepoint [14] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [15] 0 0
Change in creatinine levels as part of standard serum chemistry panel.
Timepoint [15] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [16] 0 0
Change in total protein levels as part of standard serum chemistry panel.
Timepoint [16] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [17] 0 0
Changes in total albumin levels as part of standard serum chemistry panel.
Timepoint [17] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [18] 0 0
Change in total ALP levels as part of standard serum chemistry panel.
Timepoint [18] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [19] 0 0
Change in total ALT levels as part of standard serum chemistry panel.
Timepoint [19] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [20] 0 0
Change in total AST levels as part of standard serum chemistry panel.
Timepoint [20] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [21] 0 0
Change in total bilirubin levels as part of standard serum chemistry panel.
Timepoint [21] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [22] 0 0
Change in total indirect bilirubin levels as part of standard serum chemistry panel.
Timepoint [22] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [23] 0 0
Change in total amylase levels as part of standard serum chemistry panel.
Timepoint [23] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [24] 0 0
Change in total lipase levels as part of standard serum chemistry panel.
Timepoint [24] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [25] 0 0
Change in total uric acid levels as part of standard serum chemistry panel.
Timepoint [25] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [26] 0 0
Change in total creatine kinase (CK) levels as part of standard serum chemistry panel.
Timepoint [26] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [27] 0 0
Change in total calcium levels as part of standard serum chemistry panel.
Timepoint [27] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [28] 0 0
Change in total magnesium levels as part of standard serum chemistry panel.
Timepoint [28] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [29] 0 0
Change in total lactate dehydrogenase (LDH) levels as part of standard serum chemistry panel.
Timepoint [29] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [30] 0 0
Change in total immunoglobulin (IgG) levels as part of standard serum chemistry panel.
Timepoint [30] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [31] 0 0
Change in total immunoglobulin (IgA) levels as part of standard serum chemistry panel.
Timepoint [31] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [32] 0 0
Changes in total immunoglobulin (IgE) levels as part of standard serum chemistry panel.
Timepoint [32] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [33] 0 0
Change in total immunoglobulin (IgM) levels as part of standard serum chemistry panel.
Timepoint [33] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [34] 0 0
Change in hematocrit as part of standard hematology panel.
Timepoint [34] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [35] 0 0
Change in red blood cell (RBC) counts as part of standard hematology panel.
Timepoint [35] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [36] 0 0
Change in platelet (PLT) counts as part of standard hematology panel.
Timepoint [36] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [37] 0 0
Change in white blood cell (WBC) counts as part of standard hematology panel.
Timepoint [37] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [38] 0 0
Change in neutrophil percentage as part of standard hematology panel.
Timepoint [38] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [39] 0 0
Change in lymphocyte percentage as part of standard hematology panel.
Timepoint [39] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [40] 0 0
Change in eosinophil percentage as part of standard hematology panel.
Timepoint [40] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [41] 0 0
Change in basophil percentage as part of standard hematology panel.
Timepoint [41] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [42] 0 0
Change in monocyte percentage as part of standard hematology panel.
Timepoint [42] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [43] 0 0
Change in clarity as part of a standard urinalysis panel.
Timepoint [43] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [44] 0 0
Change in specific gravity as part of a standard urinalysis panel.
Timepoint [44] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [45] 0 0
Change in pH as part of a standard urinalysis panel.
Timepoint [45] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [46] 0 0
Change in protein levels as part of a standard urinalysis panel.
Timepoint [46] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [47] 0 0
Change in glucose levels as part of a standard urinalysis panel.
Timepoint [47] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [48] 0 0
Change in ketone levels as part of a standard urinalysis panel.
Timepoint [48] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [49] 0 0
Change in blood levels as part of a standard urinalysis panel.
Timepoint [49] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [50] 0 0
Change in nitrite levels as part of a standard urinalysis panel.
Timepoint [50] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Primary outcome [51] 0 0
Change in leukocyte esterase levels as part of a standard urinalysis panel.
Timepoint [51] 0 0
Screening, day 1, day 2, day 3 and 30 days after dosing.
Secondary outcome [1] 0 0
PK assessment: Cmax (observed maximum serum concentration taken directly from the individual concentration-time curve)
Timepoint [1] 0 0
Pre-dose and post-dose at 5, 10, 20 minutes,1 and 4 hours
Secondary outcome [2] 0 0
PK assessment Tmax (Time to reach maximum serum concentration, taken directly from the individual concentration-time curve)
Timepoint [2] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days)
Secondary outcome [3] 0 0
PK assessment: t1/2 (Terminal half-life)
Timepoint [3] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days
Secondary outcome [4] 0 0
PK assessment: AUC(0-last) (Area under the serum concentration-curve from time zero to the time of last quantifiable analyte concentration)
Timepoint [4] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days
Secondary outcome [5] 0 0
PK assessment: AUC (Area under the concentration-time curve in the serum zero (pre-dose) extrapolated to infinite time)
Timepoint [5] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days
Secondary outcome [6] 0 0
PK assessment: AUC(0-24) (Area under the plasma concentration-curve)
Timepoint [6] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days
Secondary outcome [7] 0 0
PK assessment: Vz/F (Apparent volume of distribution during terminal phase)
Timepoint [7] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days
Secondary outcome [8] 0 0
PK assessment: CL/F (Apparent oral clearance estimated as dose divided by AUC)
Timepoint [8] 0 0
Pre-dose and post-dose at 5, 20 and 40 minutes, 1, 1.5, 2, 3, 4, 8,12,15,18, 36 and 48 hours and at 30 days
Secondary outcome [9] 0 0
PK assessment of urine
Timepoint [9] 0 0
Pre-dose and continuously during the following time-intervals: 0-4, 4-8, 8-12, 12-18, 18-24, 24-30, 30-36, 36-42 and 42-48 hours

Eligibility
Key inclusion criteria
* Healthy male and female of non-childbearing potential (post-menopausal or surgically sterilized) subjects of 18 to 55 years of age
* Body mass index (BMI) of 18-35
* Subjects who are non-smokers or ex-smokers who have not smoked in the last 6 months (determined by urine cotinine < 500 ng/ml, at screening visit).
Minimum age
18 Years
Maximum age
55 Years
Sex
Both males and females
Can healthy volunteers participate?
Yes
Key exclusion criteria
* History or clinical manifestations of any clinically significant medical disorder that, in the opinion of the investigator, may put the subject at risk because of participation in the study, influence the results of the study or affect the subject's ability to participate in the study.
* A history of drug or alcohol abuse.
* History of, or known significant infection including hepatitis A, B, or C, Human immunodeficiency Virus (HIV), tuberculosis (i.e., positive result for Interferon (INF)-y release assay (IGRA), QuantiFERON TB-Gold), that may put the subject at risk during participation in the study.
* Any clinically significant illness, infection, medical/surgical procedure, or trauma within 4 weeks of day 1 or planned inpatient surgery or hospitalization during the study period.
* Subjects with any history of malignancy or neoplastic disease.
* Any clinically significant abnormalities in clinical chemistry, hematology, or urinalysis results, as judged by the principal investigator.
* Subjects who have received live or attenuated vaccine in the 4 weeks prior to day 1 subjects with a disease history suggesting abnormal immune function
* Inability to communicate well with the Investigator (i.e. language problem, poor mental development or impaired cerebral function)
* Participation in any clinical study for a New Chemical Entity within the previous 16 weeks or a marketed drug clinical study within the previous 12 weeks or within 5 half- lives, whichever is the longer, before the first dose of study drug.
* Donation of 450 ml or more blood within the previous 12 weeks
* Women who are pregnant
* Males who are sexually active with a female partner of childbearing potential and who have not had a vasectomy and who do not agree to double methods of contraception with at least one barrier from day 1 for 90 days.

Study design
Purpose of the study
Treatment
Allocation to intervention
Randomised controlled trial
Procedure for enrolling a subject and allocating the treatment (allocation concealment procedures)
Methods used to generate the sequence in which subjects will be randomised (sequence generation)
Masking / blinding
Blinded (masking used)
Who is / are masked / blinded?
The people receiving the treatment/s


Intervention assignment
Parallel
Other design features
Phase
Phase 1
Type of endpoint/s
Statistical methods / analysis

Recruitment
Recruitment status
Completed
Data analysis
Reason for early stopping/withdrawal
Other reasons
Date of first participant enrolment
Anticipated
Actual
Date of last participant enrolment
Anticipated
Actual
Date of last data collection
Anticipated
Actual
Sample size
Target
Accrual to date
Final
Recruitment in Australia
Recruitment state(s)
VIC
Recruitment hospital [1] 0 0
Nucleus Network Limited - Melbourne
Recruitment postcode(s) [1] 0 0
3004 - Melbourne

Funding & Sponsors
Primary sponsor type
Commercial sector/industry
Name
Pieris Australia Pty Ltd
Address
Country

Ethics approval
Ethics application status

Summary
Brief summary
Trial website
Trial related presentations / publications
Public notes

Contacts
Principal investigator
Name 0 0
Jason Lickliter, MBBS PhD
Address 0 0
Nucleus Network
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for public queries
Name 0 0
Address 0 0
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for scientific queries

Data sharing statement
Will individual participant data (IPD) for this trial be available (including data dictionaries)?
Undecided
No/undecided IPD sharing reason/comment


What supporting documents are/will be available?

No Supporting Document Provided



Results publications and other study-related documents

No documents have been uploaded by study researchers.